Total Synthesis of Propolisbenzofuran B.
نویسندگان
چکیده
The first total synthesis of propolisbenzofuran B, a bioactive natural product isolated from honeybee propolis resin, is reported. The convergent synthesis makes use of a silicon-tether controlled oxidative ketone-ketone cross-coupling and a novel benzofuran-generating cascade reaction to deliver the core structure of the natural product from readily prepared precursors.
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ورودعنوان ژورنال:
- Chemical science
دوره 5 5 شماره
صفحات -
تاریخ انتشار 2014